SCHEMBL21190883

SCHEMBL21190883

CC(C)(C)N[S+]([O-])c1ccc(Oc2ccc(F)cc2F)c(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSPB1 P04792 2/20 0.35
BRD4 O60885 4/20 0.34
PTGS2 P35354 1/20 0.31
EPAS1 Q99814 1/20 0.31
SCN9A Q15858 1/20 0.30
LPL P06858 1/20 0.30
LIPG Q9Y5X9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19931317 0.82 HSPB1 (0.37) HSPB1BRD4PTGS2EPAS1LPL
SCHEMBL21190879 0.79 BRD4 (0.47) HSPB1BRD4PTGS2EPAS1SCN9A
SCHEMBL21904915 0.76 HSPB1 (0.39) HSPB1BRD4PTGS2LPLLIPG
SCHEMBL29533045 0.75 HSPB1 (0.39) HSPB1BRD4PTGS2LPLLIPG
SCHEMBL15069672 0.75 HSPB1 (0.39) HSPB1BRD4PTGS2LPLLIPG
SCHEMBL20155120 0.74 ALDH1A1 (0.40) HSPB1BRD4PTGS2LPLLIPG
SCHEMBL20155140 0.73 PTGS2 (0.51) HSPB1BRD4PTGS2EPAS1
SCHEMBL20268765 0.73 HSPB1 (0.63) HSPB1PTGS2
SCHEMBL31073743 0.73 HSPB1 (0.38) HSPB1BRD4PTGS2EPAS1LPL
SCHEMBL16651407 0.72 BRD4 (0.47) HSPB1BRD4PTGS2EPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed
US-9359548-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2016-06-07 US disclosed