SCHEMBL21190899

SCHEMBL21190899

CSCc1ccc(OC2CCCCC2)c(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 2/20 0.43
KMT2A Q03164 7/20 0.43
MEN1 O00255 6/20 0.43
NPY1R P25929 1/20 0.43
NPY2R P49146 1/20 0.43
THRA P10827 2/20 0.42
THRB P10828 2/20 0.42
POLB P06746 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
MAPT P10636 2/20 0.40
LMNA P02545 2/20 0.40
RECQL P46063 1/20 0.39
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GFER P55789 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
PDE4B Q07343 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21191018 0.86 SYK (0.42) CSNK2A1KMT2ANPY1RNPY2RGFER
SCHEMBL21190906 0.84 BRD4 (0.36) CSNK2A1KMT2AMEN1NPY1RNPY2R
SCHEMBL21190898 0.82 CSNK2A1 (0.48) CSNK2A1KMT2AMEN1NPY1RNPY2R
SCHEMBL21190896 0.82 THRA (0.49) CSNK2A1KMT2AMEN1NPY1RNPY2R
SCHEMBL21190894 0.78 BRD4 (0.51) CSNK2A1KMT2AMEN1NPY1RNPY2R
SCHEMBL20443015 0.78 KMT2A (0.43) CSNK2A1KMT2AMEN1NPY1RNPY2R
SCHEMBL12355729 0.76 KMT2A (0.50) CSNK2A1KMT2AMEN1NPY1RNPY2R
SCHEMBL21191023 0.75 HRH3 (0.39) KMT2ATHRATHRBL3MBTL1GFER
SCHEMBL20384189 0.75 HPGD (0.43) CSNK2A1KMT2AMEN1NPY1RNPY2R
SCHEMBL3689787 0.74 THRA (0.52) KMT2AMEN1THRATHRBPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed
US-9359548-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2016-06-07 US disclosed