SCHEMBL21190894

SCHEMBL21190894

CS(=O)(=O)Cc1ccc(OC2CCCCC2)c(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.51
THRA P10827 2/20 0.43
THRB P10828 2/20 0.43
POLB P06746 1/20 0.42
CSNK2A1 P68400 2/20 0.42
PDE4B Q07343 3/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP19A1 P11511 2/20 0.39
PTGES O14684 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
PTGS1 P23219 1/20 0.39
CYP2C19 P33261 1/20 0.39
PTGS2 P35354 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21191020 0.87 BRD4 (0.52) BRD4PDE4BPDE4APDE4CPDE4D
SCHEMBL21190903 0.85 BRD4 (0.54) BRD4
SCHEMBL21190898 0.80 CSNK2A1 (0.48) THRATHRBPOLBCSNK2A1PDE4B
SCHEMBL21190896 0.80 THRA (0.49) THRATHRBPOLBCSNK2A1PDE4B
SCHEMBL20443010 0.79 POLB (0.49) BRD4POLBMEN1KMT2ACYP19A1
SCHEMBL21190899 0.78 CSNK2A1 (0.43) THRATHRBPOLBCSNK2A1PDE4B
SCHEMBL16335601 0.77 RORC (0.47) BRD4POLBPDE4BMEN1KMT2A
SCHEMBL21191022 0.77 BRD4 (0.50) BRD4THRATHRBPDE4BPDE4A
SCHEMBL21190876 0.76 BRD4 (0.52) BRD4THRATHRBPOLBPDE4B
SCHEMBL21190895 0.76 BRD4 (0.45) BRD4CSNK2A1PDE4BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed
US-9359548-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2016-06-07 US disclosed