SCHEMBL2123165

SCHEMBL2123165

Cc1c(F)cc(Cl)c2[nH]ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.41
TNF P01375 1/20 0.39
RIPK1 Q13546 1/20 0.39
AURKA O14965 4/20 0.36
TPX2 Q9ULW0 3/20 0.36
PRKCQ Q04759 2/20 0.35
PRKCD Q05655 1/20 0.35
NR3C1 P04150 2/20 0.34
PGR P06401 2/20 0.34
NR3C2 P08235 2/20 0.34
AR P10275 2/20 0.34
AHR P35869 1/20 0.33
RHEB Q15382 1/20 0.33
AXL P30530 2/20 0.33
PRKCI P41743 2/20 0.33
CCR8 P51685 1/20 0.32
DAPK3 O43293 1/20 0.32
JAK2 O60674 1/20 0.32
PRKD3 O94806 1/20 0.32
MAP4K4 O95819 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31357988 0.81 TNF (0.46) P2RX7TNFRIPK1NR3C1PGR
SCHEMBL20939366 0.81 P2RX7 (0.42) P2RX7AURKATPX2PRKCQPRKCD
SCHEMBL24786395 0.78 TNF (0.43) P2RX7TNFRIPK1ARAHR
SCHEMBL1146475 0.78 P2RX7 (0.40) P2RX7AURKATPX2PRKCQPRKCD
SCHEMBL18876102 0.75 AURKA (0.36) TNFRIPK1AURKATPX2PRKCQ
SCHEMBL12748352 0.75 TNF (0.38) P2RX7TNFRIPK1NR3C1PGR
SCHEMBL26145363 0.74 AURKA (0.34) P2RX7AURKATPX2
SCHEMBL26145674 0.73 AURKA (0.36) P2RX7TNFRIPK1AURKATPX2
SCHEMBL24215565 0.73 TNF (0.41) P2RX7TNFRIPK1NR3C1PGR
SCHEMBL15797379 0.73 AURKA (0.58) P2RX7AURKATPX2PRKAA1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120091815-A T-type voltage-gated calcium channel enhancer 广泛研究所股份有限公司 2025-06-03 CN disclosed
EP-2444401-B1 NOVEL IMIDAZOPYRIDINE COMPOUND ONO PHARMACEUTICAL CO (JP) 2014-09-03 EP disclosed
US-8569504-B2 Imidazopyridine compound ONO PHARMACEUTICAL CO., LTD. (JP) 2013-10-29 US disclosed
EP-2444401-A1 NOVEL IMIDAZOPYRIDINE COMPOUND ONO Pharmaceutical Co., Ltd. (JP) 2012-04-25 EP disclosed
US-20120094944-A1 NOVEL IMIDAZOPYRIDINE COMPOUND ONO PHARMACEUTICAL CO., LTD. (JP) 2012-04-19 US disclosed
US-20110071146-A1 17BetaHSD Type 5 Inhibitor ASTELLAS PHARMA INC. 2011-03-24 US disclosed
US-7855225-B2 17βHSD type 5 inhibitor ASTELLAS PHARMA INC. (JP) 2010-12-21 US disclosed
US-7855225-B2 17βHSD type 5 inhibitor ASTELLAS PHARMA INC. (JP) 2010-12-21 US disclosed
US-20090181960-A1 Selective enzyme inhibitors of 17-beta-hydroxysteroid dehydrogenase (17 beta HSD); 1-[(4-bromophenyl)sulfonyl]-1H-indole-3-carboxylic acid, andanalogues; benign prostate hyperplasia; prostate cancer; acne, seborrhea, hirsutism, baldness, alopecia, precocious puberty, adrenal hypertrophy, breast cancer ASTELLAS PHARMA INC. (JP) 2009-07-16 US disclosed
US-20090181960-A1 Selective enzyme inhibitors of 17-beta-hydroxysteroid dehydrogenase (17 beta HSD); 1-[(4-bromophenyl)sulfonyl]-1H-indole-3-carboxylic acid, andanalogues; benign prostate hyperplasia; prostate cancer; acne, seborrhea, hirsutism, baldness, alopecia, precocious puberty, adrenal hypertrophy, breast cancer ASTELLAS PHARMA INC. (JP) 2009-07-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110071146-A1 17BetaHSD Type 5 Inhibitor CYP17A1, HSD17B3, HSD3B1 P2RX7 4849/4885TNF 3331/4885RIPK1 2929/4885
US-20120094944-A1 NOVEL IMIDAZOPYRIDINE COMPOUND CMA1, ACE, ALPI P2RX7 2432/4885TNF 690/4885RIPK1 3714/4885
US-20090181960-A1 Selective enzyme inhibitors of 17-beta-hydroxysteroid dehydrogenase (17 beta HSD); 1-[(4-bromophenyl)sulfonyl]-1H-indole-3-carboxylic acid, andanalogues; benign prostate hyperplasia; prostate cancer; acne, seborrhea, hirsutism, baldness, alopecia, precocious puberty, adrenal hypertrophy, breast cancer CYP17A1, HSD17B3, HSD17B1 P2RX7 4865/4885TNF 2693/4885RIPK1 2520/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.