SCHEMBL21236746

SCHEMBL21236746

CC(C)=CCOc1cc(O)c2c(=O)cc(-c3ccccc3)oc2c1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.80
EGFR P00533 1/20 0.73
RET P07949 1/20 0.73
KDR P35968 1/20 0.73
MAPT P10636 5/20 0.69
ABCB1 P08183 4/20 0.69
ABCG2 Q9UNQ0 3/20 0.67
CYP3A4 P08684 2/20 0.67
CYP2C9 P11712 2/20 0.67
CYP2C19 P33261 2/20 0.67
NPC1 O15118 1/20 0.67
TSHR P16473 1/20 0.67
CYP1A1 P04798 2/20 0.65
CYP1A2 P05177 2/20 0.65
NPSR1 Q6W5P4 1/20 0.64
LMNA P02545 1/20 0.62
KDM4E B2RXH2 2/20 0.62
MEN1 O00255 1/20 0.62
GABRP O00591 1/20 0.62
GABRD O14764 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29494586 1.00 PPARG (0.80) PPARGEGFRRETKDRMAPT
SCHEMBL4839605 0.88 PLG (0.67) PPARGMAPTABCB1ABCG2CYP3A4
SCHEMBL4056341 0.86 MAPT (0.72) PPARGEGFRRETKDRMAPT
SCHEMBL8391032 0.83 EGFR (0.74) EGFRRETKDRMAPTABCB1
SCHEMBL24882669 0.82 EGFR (0.78) PPARGEGFRRETKDRMAPT
SCHEMBL10025658 0.82 MAPT (0.77) PPARGEGFRRETKDRMAPT
SCHEMBL30376285 0.82 MAPT (1.00) PPARGEGFRRETKDRMAPT
SCHEMBL974548 0.82 MAPT (1.00) PPARGEGFRRETKDRMAPT
SCHEMBL12678185 0.81 EGFR (0.80) EGFRRETKDRMAPTABCB1
SCHEMBL22729259 0.81 MAPT (0.81) PPARGEGFRRETKDRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210038562-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING DIABETES COMPLICATIONS COMPRISING NOVEL CHRYSIN DERIVATIVE COMPOUND AS ACTIVE INGREDIENT FRONTBIO INC. (KR) 2021-02-11 US disclosed
EP-3747435-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING DIABETES COMPLICATIONS COMPRISING NOVEL CHRYSIN DERIVATIVE COMPOUND AS ACTIVE INGREDIENT FRONTBIO INC. (KR) 2020-12-09 EP disclosed
EP-3747435-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING DIABETES COMPLICATIONS COMPRISING NOVEL CHRYSIN DERIVATIVE COMPOUND AS ACTIVE INGREDIENT FRONTBIO INC. (KR) 2020-12-09 EP disclosed
WO-2019151732-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING DIABETES COMPLICATIONS COMPRISING NOVEL CHRYSIN DERIVATIVE COMPOUND AS ACTIVE INGREDIENT 한림대학교 산학협력단 2019-08-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210038562-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING DIABETES COMPLICATIONS COMPRISING NOVEL CHRYSIN DERIVATIVE COMPOUND AS ACTIVE INGREDIENT AGER, IAPP, GCG PPARG 254/4885EGFR 2350/4885RET 3120/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.