SCHEMBL2123807

SCHEMBL2123807

Cc1c(OS(=O)(=O)C(F)(F)F)ccc2c1CCN(C(=O)O)CC2C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 12/20 0.37
DRD3 P35462 9/20 0.37
DRD4 P21917 8/20 0.37
DRD1 P21728 6/20 0.37
DRD5 P21918 6/20 0.37
HTR5A P47898 1/20 0.34
HTR1D P28221 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2124391 0.88 DRD2 (0.48) DRD2DRD3DRD4DRD1DRD5
SCHEMBL2123810 0.83 DRD2 (0.36) DRD2DRD3DRD4DRD1DRD5
SCHEMBL2123254 0.82 DRD2 (0.38) DRD2DRD3DRD4DRD1DRD5
SCHEMBL2122364 0.79 ESR1 (0.39)
SCHEMBL2121244 0.79 ESR1 (0.40) DRD2DRD3DRD4DRD1DRD5
SCHEMBL3430802 0.79 DRD2 (0.36) DRD2DRD3DRD4DRD1DRD5
SCHEMBL2121801 0.77 NOTUM (0.34)
SCHEMBL2123989 0.76 SLC6A2 (0.36) DRD2
SCHEMBL2120946 0.75 ESR2 (0.44) DRD2
SCHEMBL2117067 0.74 ESR2 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443110-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING Glaxo Group Limited (GB) 2012-04-25 EP disclosed
WO-2010146105-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING GLAXO GROUP LIMITED (GB) 2010-12-23 WO disclosed