SCHEMBL3430802

SCHEMBL3430802

Cc1cc2c(cc1OS(=O)(=O)C(F)(F)F)C(C(C)(C)C)CN(C(=O)O)CC2

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.36
DRD3 P35462 6/20 0.33
DRD1 P21728 4/20 0.33
DRD4 P21917 4/20 0.33
DRD5 P21918 4/20 0.33
MTNR1B P49286 2/20 0.33
NQO2 P16083 1/20 0.33
MTNR1A P48039 1/20 0.33
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2121244 0.84 ESR1 (0.40) DRD2DRD3DRD1DRD4DRD5
SCHEMBL3430803 0.83 MEN1 (0.38) DRD2MTNR1BNQO2MTNR1ASMN1; SMN2
SCHEMBL2123807 0.79 DRD2 (0.37) DRD2DRD3DRD1DRD4DRD5
SCHEMBL2124391 0.77 DRD2 (0.48) DRD2DRD3DRD1DRD4DRD5
SCHEMBL2122587 0.77 ESR1 (0.38) DRD2DRD1ESR1ESR2SMN1; SMN2
SCHEMBL18759887 0.76 SMN1; SMN2 (0.40) MTNR1BSMN1; SMN2LMNA
SCHEMBL2123572 0.76 ESR2 (0.46) ESR2
SCHEMBL2121610 0.73 USP30 (0.34) LMNA
SCHEMBL25343893 0.73 ESR2 (0.52) DRD2ESR1ESR2
SCHEMBL29784593 0.73 ESR2 (0.52) DRD2ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010146105-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING GLAXO GROUP LIMITED (GB) 2010-12-23 WO disclosed