SCHEMBL21241205

SCHEMBL21241205

COc1cnc(N)cc1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 4/20 0.58
NOS2 P35228 4/20 0.58
NOS1 P29475 3/20 0.58
GABRP O00591 1/20 0.46
GABRD O14764 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB1 P18505 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GABRA2 P47869 1/20 0.46
GABRB2 P47870 1/20 0.46
GABRA4 P48169 1/20 0.46
GABRE P78334 1/20 0.46
GABRA6 Q16445 1/20 0.46
GABRG1 Q8N1C3 1/20 0.46
GABRG3 Q99928 1/20 0.46
GABRQ Q9UN88 1/20 0.46
P2RX3 P56373 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91466 0.83 NOS3 (0.58) NOS3NOS2NOS1GABRPGABRD
SCHEMBL29637494 0.82 NOS3 (0.44) NOS3NOS2NOS1P2RX3P2RX2
SCHEMBL29637497 0.82 NOS3 (0.44) NOS3NOS2NOS1P2RX3P2RX2
SCHEMBL2894993 0.82 NOS3 (0.44) NOS3NOS2NOS1P2RX3P2RX2
SCHEMBL23882539 0.80 NOS3 (0.50) NOS3NOS2NOS1GABRPGABRD
SCHEMBL4142773 0.77 UHRF1 (0.48) P2RX3P2RX2ALDH1A1TAAR1PDGFRB
SCHEMBL22491094 0.77 GAA (0.50) NOS3NOS2NOS1P2RX3P2RX2
SCHEMBL23068062 0.77 P2RX3 (0.43) NOS3NOS2NOS1P2RX3P2RX2
SCHEMBL27485620 0.76 NNMT (0.52) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL21223488 0.75 HSD17B10 (0.49) NOS3NOS2NOS1DHFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023056441-A1 CDK INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS INCORPORATED (US) 2023-04-06 WO disclosed
WO-2021050824-A1 CDK INHIBITORS AND THEIR USE AS PHARMACEUTICALS PRELUDE THERAPEUTICS INCORPORATED (US) 2021-03-18 WO disclosed
WO-2019149260-A1 PYRIDAZINOL COMPOUND, DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR, HERBICIDAL COMPOSITION AND USE THEREOF 青岛清原化合物有限公司 2019-08-08 WO disclosed