SCHEMBL21246342

SCHEMBL21246342

COc1cc(CNC(=O)[C@H]([C@@H](C)O)N2CC3(CCCCC3)CC2=O)cc(OC)c1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
POLB P06746 2/20 0.41
LDHA P00338 1/20 0.40
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
MAPK10 P53779 1/20 0.35
LIPG Q9Y5X9 1/20 0.35
PDE2A O00408 1/20 0.35
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21246341 0.90 LMNA (0.48) CYP3A4POLBLMNAMEN1KMT2A
SCHEMBL21246364 0.89 CYP3A4 (0.41) CYP3A4LMNATP53KDM4E
SCHEMBL21246339 0.86 PTPN1 (0.40) LMNA
SCHEMBL21246338 0.85 KMT2A (0.38) LMNATP53MEN1KMT2AKDM4E
SCHEMBL21246428 0.85 LMNA (0.48) LMNATP53MEN1KMT2AALDH1A1
SCHEMBL21246368 0.84 MAPT (0.44) POLBLMNATP53ALDH1A1NAMPT
SCHEMBL21246363 0.83 HTT (0.46) LMNAMEN1KMT2AALDH1A1TSHR
SCHEMBL21246366 0.83 THRB (0.47) CYP3A4POLBLMNAMEN1KMT2A
SCHEMBL21246365 0.83 TSHR (0.46) CYP3A4POLBMEN1KMT2AALDH1A1
SCHEMBL21246427 0.82 SLC1A2 (0.47) CYP3A4LMNAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019152688-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2019-08-08 WO disclosed