SCHEMBL21246537

SCHEMBL21246537

CC(C)(C)OC(=O)NCC(=O)N1CC2(CCCCC2)CC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
SIGMAR1 Q99720 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
EPHX1 P07099 1/20 0.34
NPFFR1 Q9GZQ6 1/20 0.34
NPFFR2 Q9Y5X5 1/20 0.34
DRD2 P14416 4/20 0.33
HDAC8 Q9BY41 1/20 0.33
KDM4E B2RXH2 2/20 0.33
LMNA P02545 2/20 0.33
EPHX2 P34913 1/20 0.33
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
P2RX7 Q99572 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21225110 0.80 GRM5 (0.32)
SCHEMBL3078624 0.79 BUB1 (0.37) EPHX1KDM4EHPGD
SCHEMBL3733841 0.77 KDM1A (0.38) KDM4EHPGD
SCHEMBL25238948 0.74 KDM1A (0.38) MEN1KMT2AKDM4EHPGD
SCHEMBL21225630 0.74 ITGB3 (0.40)
SCHEMBL21225628 0.74 ITGB3 (0.40)
SCHEMBL21246539 0.73 ITGB3 (0.38) HSD17B10
SCHEMBL24569354 0.71 KDM1A (0.39) KDM4EMAPT
Hydrochloric Acid SCHEMBL21225114 0.70 GRM5 (0.33) ALDH1A1KDM4E
SCHEMBL11464909 0.69 SMN1; SMN2 (0.36) ALDH1A1MEN1KMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019152688-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2019-08-08 WO disclosed