SCHEMBL21246539

SCHEMBL21246539

CC(C)(C)OC(=O)N[C@@H](CCC(N)=O)C(=O)N1CC2(CCCCC2)CC1=O

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.38
ITGA2B P08514 10/20 0.38
PLG P00747 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CTSK P43235 1/20 0.33
HSD17B10 Q99714 1/20 0.32
CTSL P07711 1/20 0.32
SUV39H2 Q9H5I1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21225630 0.91 ITGB3 (0.40) ITGB3ITGA2BCTSK
SCHEMBL21225628 0.91 ITGB3 (0.40) ITGB3ITGA2BCTSK
SCHEMBL21225293 0.84 CCKBR (0.35)
SCHEMBL21225289 0.84 CCKBR (0.35)
SCHEMBL21246541 0.82 ITGB3 (0.44) ITGB3ITGA2BCTSL
Hydrochloric Acid SCHEMBL21224547 0.75 ALOX15 (0.35)
Hydrochloric Acid SCHEMBL21224546 0.75 ALOX15 (0.35)
SCHEMBL21246537 0.73 ALDH1A1 (0.38) HSD17B10
SCHEMBL6809194 0.72 TSHR (0.41) ITGB3ITGA2BCTSKCTSL
SCHEMBL23845318 0.70 CYP1A2 (0.45) CTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019152688-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2019-08-08 WO disclosed