SCHEMBL21246887

SCHEMBL21246887

OC(CNCCCCc1ccccc1)CNc1c[nH]c2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PRMT1 Q99873 1/20 0.44
POLB P06746 1/20 0.44
HTR2A P28223 1/20 0.43
SIGMAR1 Q99720 6/20 0.42
ADRB2 P07550 2/20 0.42
ADRB1 P08588 2/20 0.42
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ADRB3 P13945 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21246885 0.81 ALDH1A1 (0.51) SIGMAR1ADRB2ADRB1ADRB3
SCHEMBL28552086 0.80 POLB (0.45) PRMT1POLBHTR2ASIGMAR1
SCHEMBL28548618 0.80 ADRB3 (0.52) HTR2ASIGMAR1ADRB2ADRB1ADRB3
SCHEMBL21259419 0.73 CYP2D6 (0.46) ADRB2ADRB1ADRB3
SCHEMBL7297780 0.71 ADRB3 (0.68) ADRB2ADRB1ADRB3
SCHEMBL7285328 0.70 ADRB3 (0.67) ADRB2ADRB1ADRB3
SCHEMBL7296273 0.70 ADRB3 (0.67) ADRB2ADRB1ADRB3
SCHEMBL6534491 0.70 SLC2A1 (0.55)
SCHEMBL6534493 0.70 SLC2A1 (0.55)
SCHEMBL2278702 0.69 KDR (0.52) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019153216-A1 SUBSTITUTED ARYLAMINO ALCOHOL COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 北京梅尔森医药技术开发有限公司 2019-08-15 WO claimed
CN-108299279-B Substituted arylaminol compounds, methods of making, and uses thereof 北京梅尔森医药技术开发有限公司 2021-03-23 CN disclosed
WO-2019153216-A1 SUBSTITUTED ARYLAMINO ALCOHOL COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 北京梅尔森医药技术开发有限公司 2019-08-15 WO disclosed