Tetraxetan

Tetraxetan

SCHEMBL21248095

NC(N)=O.O=C(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1

nearest known ligand 0.83

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.56
KDM4E B2RXH2 2/20 0.44
SLC6A9 P48067 1/20 0.43
S1PR1 P21453 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
ALOX15 P16050 1/20 0.36
ALDH1A1 P00352 2/20 0.36
STAT6 P42226 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3503521 0.91 HSD17B10 (0.64) HSD17B10KDM4ESLC6A9S1PR1ALOX15
Tetraxetan SCHEMBL2017956 0.91 HSD17B10 (0.64) HSD17B10KDM4ESLC6A9S1PR1ALOX15
Tetraxetan SCHEMBL18018 0.91 HSD17B10 (0.64) HSD17B10KDM4ESLC6A9S1PR1ALOX15
SCHEMBL6744121 0.91 HSD17B10 (0.64) HSD17B10KDM4ESLC6A9S1PR1ALOX15
SCHEMBL321989 0.91 HSD17B10 (0.64) HSD17B10KDM4ESLC6A9S1PR1ALOX15
Tetraxetan SCHEMBL2635294 0.91 HSD17B10 (0.64) HSD17B10KDM4ESLC6A9S1PR1ALOX15
SCHEMBL6848102 0.91 HSD17B10 (0.64) HSD17B10KDM4ESLC6A9S1PR1ALOX15
SCHEMBL173508 0.91 HSD17B10 (0.64) HSD17B10KDM4ESLC6A9S1PR1ALOX15
SCHEMBL3660521 0.91
SCHEMBL15043622 0.90 KDM4E (0.58) HSD17B10KDM4ESLC6A9ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11813340-B2 PSMA targeted radiohalogenated urea-polyaminocarboxylates for cancer radiotherapy THE JOHNS HOPKINS UNIVERSITY (US) 2023-11-14 US disclosed
US-20210220493-A1 PSMA TARGETED RADIOHALOGENATED UREA-POLYAMINOCARBOXYLATES FOR CANCER RADIOTHERAPY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-07-22 US disclosed
EP-3749653-A1 PSMA TARGETED RADIOHALOGENATED UREA-POLYAMINOCARBOXYLATES FOR CANCER RADIOTHERAPY The Johns Hopkins University (US) 2020-12-16 EP disclosed
CN-112020497-A PSMA-targeted radiohalogenated urea-polyaminocarboxylates for cancer radiotherapy 约翰霍普金斯大学 2020-12-01 CN disclosed
WO-2019157037-A1 PSMA TARGETED RADIOHALOGENATED UREA-POLYAMINOCARBOXYLATES FOR CANCER RADIOTHERAPY THE JOHNS HOPKINS UNIVERSITY (US) 2019-08-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210220493-A1 PSMA TARGETED RADIOHALOGENATED UREA-POLYAMINOCARBOXYLATES FOR CANCER RADIOTHERAPY PSMA1, PSMA3, PSMA2 HSD17B10 3973/4885KDM4E 824/4885SLC6A9 1624/4885
US-11813340-B2 PSMA targeted radiohalogenated urea-polyaminocarboxylates for cancer radiotherapy PSMA1, PSMA3, PSMA2 HSD17B10 3973/4885KDM4E 824/4885SLC6A9 1624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.