SCHEMBL21273155

SCHEMBL21273155

COc1ccc(-n2c(Cl)cc3c(=O)[nH]cnc32)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.46
BRD9 Q9H8M2 3/20 0.43
SRC P12931 1/20 0.41
MAP3K11 Q16584 4/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
TNF P01375 1/20 0.39
LITAF Q99732 1/20 0.39
USP7 Q93009 1/20 0.38
LMNA P02545 1/20 0.36
MCHR1 Q99705 1/20 0.36
CMA1 P23946 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21273193 0.90 USP7 (0.48) CYP2C9SRCUSP7MAPTPKM
SCHEMBL21273091 0.80 PARP1 (0.49) KMT2AMAPTALDH1A1
SCHEMBL21272834 0.78 PARP1 (0.47) KMT2AMAPTALDH1A1
SCHEMBL21273055 0.78 PARP1 (0.39) KMT2AGAALMNAMAPTALDH1A1
SCHEMBL20971266 0.78 ALDH1A1 (0.50) SRCKMT2AMAPK1LMNAMAPT
SCHEMBL19692092 0.78 SRC (0.43) CYP2C9BRD9SRCMAP3K11KMT2A
SCHEMBL21273152 0.77 ENPP1 (0.41) CYP2C9BRD9KMT2AGAAMAPK1
SCHEMBL21272804 0.75 PIM1 (0.43) KMT2AGAAUSP7LMNAMAPT
SCHEMBL23754625 0.74 PIK3CD (0.37) KMT2AUSP7ALDH1A1
SCHEMBL23754618 0.74 CYP11B2 (0.41) USP7MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4026832-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 Almac Discovery Limited (GB) 2022-07-13 EP disclosed
US-10766903-B2 Piperidine derivatives as inhibitors of ubiquitin specific protease 7 ALMAC DISCOVERY LIMITED (GB) 2020-09-08 US disclosed
US-20190256518-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 GENETECH, INC. 2019-08-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190256518-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 USP7, USP5, UBA7 CYP2C9 4240/4885BRD9 710/4885SRC 4165/4885
US-10766903-B2 Piperidine derivatives as inhibitors of ubiquitin specific protease 7 USP7, USP5, UBA7 CYP2C9 4240/4885BRD9 710/4885SRC 4165/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.