SCHEMBL21274019

SCHEMBL21274019

O=[N+]([O-])c1ccc(S(=O)(=O)OCCc2cc(F)ccc2F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPB1 P04792 4/20 0.43
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
KCNJ1 P48048 1/20 0.39
KCNH2 Q12809 1/20 0.39
ALDH1A1 P00352 3/20 0.38
HIF1A Q16665 1/20 0.38
POLB P06746 3/20 0.38
MAPT P10636 3/20 0.38
HTT P42858 2/20 0.38
HPGD P15428 1/20 0.37
RIPK1 Q13546 1/20 0.37
SLC29A1 Q99808 1/20 0.37
GAA P10253 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21274133 0.82 HSPB1 (0.41) HSPB1PSEN1PSEN2APH1BNCSTN
SCHEMBL30865768 0.77 CA1 (0.53) ALDH1A1POLBHTTCA12CA1
SCHEMBL693396 0.76 TSHR (0.51) KCNJ1KCNH2CA12CA1CA2
SCHEMBL21284573 0.76 HSPB1 (0.42) HSPB1KCNJ1KCNH2ALDH1A1HIF1A
SCHEMBL19127566 0.74 CA1 (0.47) KCNH2ALDH1A1CA12CA1CA2
SCHEMBL368915 0.74 CA1 (0.52) ALDH1A1MAPTCA12CA1CA2
SCHEMBL26181061 0.73 HSD11B1 (0.44) ALDH1A1HTTHPGDGAACA1
SCHEMBL29263722 0.73 PSEN1 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2012983 0.73 KMT2A (0.45) ALDH1A1HIF1AMAPTHTTGAA
SCHEMBL10615596 0.73 CA1 (0.48) ALDH1A1POLBMAPTHTTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019158634-A1 DEUTERATED DERIVATIVES OF 9-(2,5-DIFLUOROPHENETHYL)-4-ETHYL-2-METHYL-1-OXA-4,9-DIAZASPIRO[5.5]UNDECAN-3-ONE ESTEVE PHARMACEUTICALS, S.A. (ES) 2019-08-22 WO disclosed