SCHEMBL21284573

SCHEMBL21284573

O=[N+]([O-])c1ccc(S(=O)OCCc2cc(F)ccc2F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPB1 P04792 6/20 0.42
ALDH1A1 P00352 2/20 0.37
HIF1A Q16665 1/20 0.37
SLC29A1 Q99808 1/20 0.36
RIPK1 Q13546 1/20 0.36
KCNJ1 P48048 1/20 0.36
KCNH2 Q12809 1/20 0.36
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
POLB P06746 2/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.35
ATM Q13315 1/20 0.35
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21274019 0.76 HSPB1 (0.43) HSPB1ALDH1A1HIF1ASLC29A1RIPK1
SCHEMBL1847209 0.75 LOXL2 (0.42) HSPB1ALDH1A1KCNH2MAPTSMN1; SMN2
SCHEMBL23998043 0.69 ACHE (0.45) ALDH1A1MAPTPOLBMAPK1HTT
SCHEMBL12354045 0.66 HSPB1 (0.44) HSPB1ALDH1A1TDP1LMNA
SCHEMBL25263151 0.66 ALDH1A1 (0.44) ALDH1A1HIF1AMAPTMEN1KMT2A
SCHEMBL15778954 0.66 S1PR4 (0.57) ALDH1A1RIPK1MAPTMEN1KMT2A
SCHEMBL31156747 0.66 ALDH1A1 (0.55) ALDH1A1HIF1AMAPTMEN1KMT2A
SCHEMBL18041343 0.66 ALDH1A1 (0.55) ALDH1A1HIF1AMAPTMEN1KMT2A
SCHEMBL15076454 0.65 ALDH1A1 (0.58) HSPB1ALDH1A1HIF1AMAPTMEN1
SCHEMBL16197191 0.65 ALDH1A1 (0.53) ALDH1A1HIF1AMAPTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019158634-A1 DEUTERATED DERIVATIVES OF 9-(2,5-DIFLUOROPHENETHYL)-4-ETHYL-2-METHYL-1-OXA-4,9-DIAZASPIRO[5.5]UNDECAN-3-ONE ESTEVE PHARMACEUTICALS, S.A. (ES) 2019-08-22 WO disclosed