SCHEMBL2128776

SCHEMBL2128776

CC1(C)COc2c(-c3cc(F)c[nH]c3=O)cc(C=Cc3ccc(NS(C)(=O)=O)cc3)cc21

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
ALOX5 P09917 2/20 0.34
PTGS1 P23219 2/20 0.34
PTGS2 P35354 2/20 0.34
TDP2 O95551 1/20 0.33
PIP4K2A P48426 4/20 0.32
PIP4K2B P78356 3/20 0.32
PIP4K2C Q8TBX8 1/20 0.32
NR3C2 P08235 4/20 0.32
PADI4 Q9UM07 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1542782 1.00 CYP3A4 (0.37) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL2128431 0.85 CYP3A4 (0.49) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL1543810 0.85 CYP3A4 (0.49) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL725831 0.80 ALOX5 (0.34) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL725832 0.80 ALOX5 (0.34) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL2745734 0.79 CYP3A4 (0.38) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL2745732 0.79 CYP3A4 (0.38) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL1542617 0.74 CYP3A4 (0.59) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL2127703 0.74 CYP3A4 (0.59) CYP3A4ALOX5PTGS1PTGS2TDP2
SCHEMBL2128114 0.74 CYP3A4 (0.40) CYP3A4TDP2PIP4K2APIP4K2BPIP4K2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307372-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2012-04-25 EP claimed
US-20100021423-A1 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC 2010-01-28 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100021423-A1 Heterocyclic antiviral compounds POLR2A, RRM2B, RRP1B CYP3A4 528/4885ALOX5 3399/4885PTGS1 1761/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.