SCHEMBL21289752

SCHEMBL21289752

Oc1cc(-c2ccccn2)ccc1-c1ccccc1-c1cc(CCc2ccc(-c3ccccn3)cc2)cc(CCc2ccc(-c3ccccn3)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.42
BRS3 P32247 4/20 0.41
FFAR1 O14842 1/20 0.41
HCAR2 Q8TDS4 1/20 0.40
NR1I2 O75469 1/20 0.39
NMBR P28336 1/20 0.39
GRPR P30550 1/20 0.39
KCNH2 Q12809 1/20 0.39
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
HRH3 Q9Y5N1 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
FAAH O00519 1/20 0.36
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25100913 0.91 PDK2 (0.37) PDK2BRS3FFAR1HCAR2NR1I2
SCHEMBL25100939 0.90 WNT3A (0.39) PDK2BRS3FFAR1HCAR2NR1I2
SCHEMBL25100912 0.89 PDK2 (0.38) PDK2BRS3FFAR1HCAR2NR1I2
SCHEMBL25100916 0.89 AR (0.42) PDK2BRS3FFAR1HCAR2CA12
SCHEMBL25100884 0.88 BRS3 (0.39) PDK2BRS3FFAR1HCAR2NR1I2
SCHEMBL21290196 0.88 BRS3 (0.44) PDK2BRS3FFAR1HCAR2NR1I2
SCHEMBL26550027 0.87 FFAR1 (0.44) PDK2BRS3FFAR1HCAR2NR1I2
SCHEMBL21289804 0.87 L3MBTL1 (0.41) BRS3FFAR1HCAR2FAAHCES1
SCHEMBL21290404 0.86 FFAR1 (0.43) PDK2BRS3FFAR1HCAR2NR1I2
SCHEMBL21290071 0.86 FFAR1 (0.43) PDK2BRS3FFAR1HCAR2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed