SCHEMBL21290196

SCHEMBL21290196

c1ccc(-c2ccc(CCc3cc(CCc4ccc(-c5ccccn5)cc4)cc(-c4ccccc4-c4ccc(-c5ccccn5)cc4)c3)cc2)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 4/20 0.44
NR1I2 O75469 1/20 0.44
NMBR P28336 1/20 0.44
GRPR P30550 1/20 0.44
KCNH2 Q12809 1/20 0.44
HCAR2 Q8TDS4 1/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
FFAR1 O14842 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21290207 0.97 BRS3 (0.44) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL23487554 0.94 FFAR1 (0.45) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL29306772 0.93 GRM5 (0.41) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL26550027 0.91 FFAR1 (0.44) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL14268241 0.90 BRS3 (0.50) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL21290071 0.89 FFAR1 (0.43) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL21290404 0.89 FFAR1 (0.43) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL25100883 0.89 HCAR2 (0.41) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL21290093 0.89 TGFBR1 (0.44) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL21289814 0.89 CYP11B1 (0.46) BRS3NR1I2NMBRGRPRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed