SCHEMBL21289928

SCHEMBL21289928

COc1cc(-c2ccc(-c3ccccc3-c3cc(CCc4ccc(-c5ccc(C)cn5)cc4)cc(CCc4ccc(-c5ccc(C)cn5)cc4)c3)cc2)ncc1C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 5/20 0.38
FYN P06241 2/20 0.36
CYP11B1 P15538 3/20 0.35
CYP11B2 P19099 3/20 0.35
CYP3A4 P08684 1/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
KDM1A O60341 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SYK P43405 2/20 0.34
PTAFR P25105 2/20 0.33
GAK O14976 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21289929 0.89 BRS3 (0.39) BRS3SYK
SCHEMBL23956201 0.89 NPC1 (0.40) FYNCYP3A4KDM1AMAPTNPC1
SCHEMBL25100917 0.86 CYP11B1 (0.36) BRS3FYNCYP11B1CYP11B2CYP3A4
SCHEMBL21290192 0.85 BRS3 (0.38) BRS3CYP11B1CYP11B2CYP3A4KDM1A
SCHEMBL25100892 0.84 PTGS2 (0.35) BRS3CYP11B1CYP11B2CYP3A4
SCHEMBL25100598 0.84 CYP11B1 (0.42) BRS3CYP11B1CYP11B2CYP3A4
SCHEMBL25100886 0.83 MC4R (0.38) BRS3FYNCYP11B1CYP11B2CYP3A4
SCHEMBL25100560 0.82 HCRTR1 (0.36) BRS3MAPTL3MBTL1SYK
SCHEMBL25100532 0.81 CYP11B1 (0.42) BRS3CYP11B1CYP11B2CYP3A4
SCHEMBL25100925 0.81 CYP11B1 (0.42) BRS3CYP11B1CYP11B2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed