SCHEMBL21290192

SCHEMBL21290192

Cc1ccc(-c2ccc(CCc3cc(CCc4ccc(-c5ccc(C)cn5)cc4)cc(-c4ccccc4-c4ccc(-c5cc(O)c(C)cn5)cc4)c3)cc2)nc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 8/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
NFKB1 P19838 1/20 0.38
MAPK1 P28482 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
CYP3A4 P08684 2/20 0.36
P2RX7 Q99572 1/20 0.35
MAPT P10636 1/20 0.34
STAT3 P40763 1/20 0.34
ATM Q13315 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
CYP2A6 P11509 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21290195 0.89 BRS3 (0.40) BRS3
SCHEMBL23956165 0.88 CYP3A4 (0.40) NPC1RAB9ASMN1; SMN2TP53MAPK1
SCHEMBL25100887 0.86 RAB9A (0.42) BRS3NPC1RAB9ASMN1; SMN2TP53
SCHEMBL25100598 0.85 CYP11B1 (0.42) BRS3CYP11B1CYP11B2CYP3A4CYP2A6
SCHEMBL21289928 0.85 BRS3 (0.38) BRS3NPC1RAB9ACYP11B1CYP11B2
SCHEMBL25100532 0.83 CYP11B1 (0.42) BRS3CYP11B1CYP11B2CYP3A4CYP2A6
SCHEMBL25100925 0.83 CYP11B1 (0.42) BRS3CYP11B1CYP11B2CYP3A4CYP2A6
SCHEMBL21290225 0.83 CYP11B1 (0.38) BRS3CYP11B1CYP11B2CYP3A4P2RX7
SCHEMBL21289765 0.82 PDK1 (0.40) BRS3ESR1ESR2
SCHEMBL25100939 0.82 WNT3A (0.39) BRS3NPC1RAB9ASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed