SCHEMBL21290146

SCHEMBL21290146

COc1cc(-c2ccc(-c3ccccc3Br)cn2)ccc1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.51
KMO O15229 1/20 0.44
DHFR P00374 1/20 0.44
KIT P10721 1/20 0.42
S1PR1 P21453 5/20 0.42
FYN P06241 3/20 0.40
PDE4D Q08499 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
NFKB1 P19838 1/20 0.38
MAPK1 P28482 1/20 0.38
NFKB2 Q00653 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21721927 0.85 NPC1 (0.48) KDM1AL3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL23956242 0.84 KDM1A (0.51) KDM1AKMODHFRKITFYN
SCHEMBL21290360 0.81 NPC1 (0.42) KDM1ADHFRKITS1PR1PDE4D
SCHEMBL21290361 0.81 POLB (0.43) KDM1AKITS1PR1FYNL3MBTL1
SCHEMBL21290349 0.80 KDM1A (0.58) KDM1AKMODHFRS1PR1FYN
SCHEMBL21290362 0.80 TP53 (0.53) KDM1AFYNMAPT
SCHEMBL19933811 0.78 HSD17B1 (0.53) KDM1AL3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL23239937 0.78 KDM1A (0.47) KDM1AKMONPC1RAB9ASMN1; SMN2
SCHEMBL19933810 0.78 ALDH1A1 (0.50) L3MBTL1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL20068872 0.76 MAPK1 (0.52) L3MBTL1NPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed