SCHEMBL21290360

SCHEMBL21290360

COc1cc(-c2ccc(-c3ccccc3Br)cc2)ncc1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
IDO1 P14902 4/20 0.41
TDO2 P48775 4/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 1/20 0.40
DYRK1A Q13627 1/20 0.39
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
POLB P06746 1/20 0.38
PDE4D Q08499 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DHFR P00374 1/20 0.37
PLK1 P53350 1/20 0.36
KDM1A O60341 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21290146 0.81 KDM1A (0.51) NPC1RAB9AL3MBTL1ALDH1A1MAPK1
SCHEMBL23956221 0.80 TGFBR1 (0.42) NPC1RAB9AIDO1TDO2L3MBTL1
SCHEMBL23956201 0.80 NPC1 (0.40) NPC1RAB9AIDO1TDO2ALDH1A1
SCHEMBL21290149 0.80 IDO1 (0.48) NPC1RAB9AIDO1TDO2L3MBTL1
SCHEMBL18015459 0.78 MAPK1 (0.52) NPC1RAB9AL3MBTL1ALDH1A1MAPK1
SCHEMBL21290347 0.77 IDO1 (0.54) NPC1RAB9AIDO1TDO2L3MBTL1
SCHEMBL20075600 0.77 ALDH1A1 (0.50) NPC1RAB9AL3MBTL1ALDH1A1MAPK1
SCHEMBL21290159 0.76 CXCL12 (0.48) NPC1RAB9AIDO1TDO2L3MBTL1
SCHEMBL23956220 0.75 MC4R (0.39) NPC1RAB9AIDO1TDO2DYRK1A
SCHEMBL18015452 0.75 LDHA (0.41) NPC1RAB9AIDO1TDO2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed