SCHEMBL25100883

SCHEMBL25100883

Oc1ccnc(-c2ccc(-c3ccccc3-c3cc(CCc4ccc(-c5ccccn5)cc4)cc(CCc4ccc(-c5ccccn5)cc4)c3)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.41
FFAR1 O14842 2/20 0.41
BRS3 P32247 4/20 0.38
NR1I2 O75469 1/20 0.38
NMBR P28336 1/20 0.38
GRPR P30550 1/20 0.38
KCNH2 Q12809 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
MET P08581 1/20 0.37
RET P07949 2/20 0.37
PDK2 Q15119 1/20 0.36
KDM1A O60341 1/20 0.36
ABL1 P00519 1/20 0.36
ABCB1 P08183 1/20 0.36
BCR P11274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21290196 0.89 BRS3 (0.44) HCAR2FFAR1BRS3NR1I2NMBR
SCHEMBL23956249 0.87 NPC1 (0.45) NPC1RAB9ARETPDK2KDM1A
SCHEMBL21290207 0.87 BRS3 (0.44) HCAR2FFAR1BRS3NR1I2NMBR
SCHEMBL29306772 0.86 GRM5 (0.41) HCAR2FFAR1BRS3NR1I2NMBR
SCHEMBL21290093 0.85 TGFBR1 (0.44) HCAR2FFAR1BRS3NR1I2NMBR
SCHEMBL23487554 0.84 FFAR1 (0.45) HCAR2FFAR1BRS3NR1I2NMBR
SCHEMBL21289752 0.84 PDK2 (0.42) HCAR2FFAR1BRS3NR1I2NMBR
SCHEMBL21290226 0.83 TGFBR1 (0.43) HCAR2FFAR1BRS3NR1I2NMBR
SCHEMBL21289816 0.82 TGFBR1 (0.44) HCAR2FFAR1BRS3NR1I2NMBR
SCHEMBL21290195 0.82 BRS3 (0.40) HCAR2FFAR1BRS3NR1I2NMBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed