SCHEMBL21290367

SCHEMBL21290367

Fc1ccc(-c2ccc(Br)cn2)c(F)n1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
SPR P35270 1/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
NFKB1 P19838 1/20 0.33
RAB9A P51151 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GRM5 P41594 1/20 0.31
PLAU P00749 1/20 0.30
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
GBA1 P04062 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19248524 0.81 MAPT (0.35) NPC1GRM5
SCHEMBL19072766 0.76 NPSR1 (0.40) ALOX5APFEN1RAB9AKDM4E
SCHEMBL18932589 0.76
SCHEMBL18944253 0.75 PTGS2 (0.36) ALOX5APFEN1
SCHEMBL13713457 0.73 ADORA2A (0.35) ALOX5APFEN1NPC1GAARAB9A
SCHEMBL13713452 0.73 FEN1 (0.37) ALOX5APFEN1GRM5
SCHEMBL503341 0.72 ALOX5AP (0.43) ALOX5APFEN1SPRNPC1GAA
SCHEMBL38614 0.71 FEN1 (0.47) ALOX5APFEN1NPC1GAANFKB1
SCHEMBL114154 0.71
SCHEMBL4316048 0.71 KDM4E (0.43) KDM4EALDH1A1PLAUADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed