SCHEMBL21295722

SCHEMBL21295722

[c]1ccc2oc(-c3cccnc3)cc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 6/20 0.42
KDM4E B2RXH2 4/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
PPARG P37231 1/20 0.41
CYP1A2 P05177 4/20 0.41
CYP1A1 P04798 1/20 0.41
PRKDC P78527 1/20 0.41
CYP1B1 Q16678 1/20 0.41
PGR P06401 1/20 0.41
CYP2C19 P33261 6/20 0.40
CYP2D6 P10635 5/20 0.40
CYP2C9 P11712 5/20 0.40
CYP19A1 P11511 1/20 0.40
CYP3A4 P08684 5/20 0.40
CYP2E1 P05181 3/20 0.40
CYP2B6 P20813 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 2/20 0.40
PIM1 P11309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21295874 0.88 CYP2A6 (0.42) CYP2A6KDM4EKMT2AMEN1PPARG
SCHEMBL16720104 0.81 GSK3B (0.41) CYP1A2CYP1A1CYP1B1CYP19A1MAOB
SCHEMBL1927674 0.81 MAOB (0.53) KDM4ECYP1A2CYP1A1CYP1B1CYP19A1
SCHEMBL29993564 0.80 MAOB (0.54) CYP2A6KDM4EKMT2AMEN1CYP1A2
SCHEMBL2960606 0.80 MAOB (0.54) CYP2A6KDM4EKMT2AMEN1CYP1A2
SCHEMBL15867533 0.79 CYP19A1 (0.51) CYP2A6KDM4EKMT2AMEN1PPARG
SCHEMBL30461597 0.76 CYP2A6 (0.47) CYP2A6KDM4EKMT2AMEN1PPARG
SCHEMBL16720144 0.75 HDAC6 (0.48) KMT2AMEN1CYP1A2CYP1A1CYP1B1
SCHEMBL16719694 0.75 GABRP (0.48) CYP1A2CYP1A1PRKDCCYP1B1MAOA
SCHEMBL2184612 0.73 ALDH1A1 (0.66) KDM4EKMT2AMEN1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311844-B Triazine compound, method for producing same, and organic electroluminescent element containing same as constituent component 东曹株式会社 2021-07-20 CN disclosed
CN-112912372-A Cyclic azine compound, material for organic electroluminescent element, electron transport material for organic electroluminescent element, and organic electroluminescent element 东曹株式会社 2021-06-04 CN disclosed
WO-2020085319-A1 CYCLIC AZINE COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENTS, ELECTRON TRANSPORT MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENTS, AND ORGANIC ELECTROLUMINESCENT ELEMENT 東ソー株式会社 2020-04-30 WO disclosed
WO-2019163959-A1 CYCLIC AZINE COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCNET ELEMENT, AND ELECTRON-TRANSPORTING MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT 東ソー株式会社 2019-08-29 WO disclosed