SCHEMBL21295784

SCHEMBL21295784

[c]1ccc2ccoc2c1-c1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.42
CYP2A6 P11509 5/20 0.42
CYP3A4 P08684 2/20 0.42
CYP1A2 P05177 1/20 0.42
CHRNB2 P17787 1/20 0.41
CHRNA5 P30532 1/20 0.41
CHRNA4 P43681 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TSHR P16473 2/20 0.41
SMN1; SMN2 Q16637 5/20 0.40
TP53 P04637 4/20 0.40
PPARA Q07869 3/20 0.38
HPGD P15428 4/20 0.38
HSD17B10 Q99714 4/20 0.38
MAPT P10636 4/20 0.38
KDM4E B2RXH2 3/20 0.38
LMNA P02545 2/20 0.38
ALOX15 P16050 2/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21295724 0.82 DYRK1A (0.41) ALDH1A1NPC1RAB9ATSHRSMN1; SMN2
SCHEMBL21295775 0.80 HTR1A (0.34) ALDH1A1CYP1A2TSHRTP53HSD17B10
SCHEMBL21295856 0.77 CYP2A6 (0.41) ALDH1A1CYP2A6CYP3A4CYP1A2CHRNB2
SCHEMBL6613858 0.74 CYP11B1 (0.50) ALDH1A1CYP2A6CYP3A4CYP1A2NPC1
SCHEMBL21295964 0.72 TP53 (0.40) ALDH1A1CYP2A6CYP1A2NPC1RAB9A
SCHEMBL21296168 0.71 CYP2A6 (0.45) ALDH1A1CYP2A6CYP3A4CYP1A2NPC1
SCHEMBL21295725 0.69 ALDH1A1 (0.52) ALDH1A1CYP2A6CYP3A4CYP1A2CHRNB2
SCHEMBL21297628 0.69 ALDH1A1 (0.42) ALDH1A1CYP2A6CYP3A4CYP1A2CHRNB2
SCHEMBL23071560 0.68 CYP2A6 (0.50) ALDH1A1CYP2A6CYP3A4CYP1A2SMN1; SMN2
SCHEMBL21295780 0.68 NUDT1 (0.43) ALDH1A1CYP2A6CYP3A4CYP1A2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311844-B Triazine compound, method for producing same, and organic electroluminescent element containing same as constituent component 东曹株式会社 2021-07-20 CN disclosed
CN-112912372-A Cyclic azine compound, material for organic electroluminescent element, electron transport material for organic electroluminescent element, and organic electroluminescent element 东曹株式会社 2021-06-04 CN disclosed
WO-2020085319-A1 CYCLIC AZINE COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENTS, ELECTRON TRANSPORT MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENTS, AND ORGANIC ELECTROLUMINESCENT ELEMENT 東ソー株式会社 2020-04-30 WO disclosed
WO-2019163959-A1 CYCLIC AZINE COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCNET ELEMENT, AND ELECTRON-TRANSPORTING MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT 東ソー株式会社 2019-08-29 WO disclosed