SCHEMBL21296833

SCHEMBL21296833

CC(=O)Oc1cn[nH]c1-c1ccccc1Nc1ccc(OCCN2CCCCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.47
ESR2 Q92731 1/20 0.46
SYK P43405 9/20 0.45
JAK2 O60674 8/20 0.45
BRD4 O60885 1/20 0.44
JAK1 P23458 1/20 0.44
HDAC1 Q13547 1/20 0.44
HRH3 Q9Y5N1 2/20 0.44
LTA4H P09960 1/20 0.44
HRH2 P25021 1/20 0.44
PSMB1 P20618 1/20 0.43
PSMB5 P28074 1/20 0.43
PSMB2 P49721 1/20 0.43
EGFR P00533 1/20 0.43
TGFBR1 P36897 1/20 0.43
CLK2 P49760 1/20 0.43
CLK3 P49761 1/20 0.43
DYRK1A Q13627 1/20 0.43
JAK3 P52333 1/20 0.43
PTK2 Q05397 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21296835 0.88 ESR1 (0.50) ESR1ESR2BRD4JAK1HDAC1
SCHEMBL21296799 0.81 ESR1 (0.47) ESR1ESR2JAK2BRD4JAK1
SCHEMBL21296780 0.79 ADRA1D (0.54) BRD4JAK1HDAC1LTA4HPSMB1
SCHEMBL21296795 0.76 MCHR1 (0.50) ESR1ESR2BRD4JAK1HDAC1
SCHEMBL21305117 0.74 LTA4H (0.44) ESR1HRH3LTA4HPSMB1PSMB5
SCHEMBL21296769 0.74 MCHR1 (0.51) BRD4JAK1HDAC1HRH3LTA4H
SCHEMBL21296831 0.74 MCHR1 (0.51) BRD4JAK1HDAC1HRH3LTA4H
SCHEMBL21296811 0.73 MCHR1 (0.49) ESR1BRD4JAK1HDAC1HRH3
SCHEMBL21296760 0.72 MCHR1 (0.50) BRD4JAK1HDAC1HRH3LTA4H
SCHEMBL7332024 0.71 ESR1 (0.73) ESR1ESR2HRH3LTA4HPSMB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019165158-A1 IL-6 INHIBITORS AND METHODS OF TREATMENT UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2019-08-29 WO disclosed