SCHEMBL21299993

SCHEMBL21299993

COC(OC)c1ccc(C(C)(C)N)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.42
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31
AOC3 Q16853 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL799991 0.82 TSHR (0.44) ALDH1A1TSHRMAPK1TDP1
SCHEMBL21300009 0.81 CYP2C9 (0.33)
SCHEMBL20746752 0.81
SCHEMBL11393154 0.80 PDE2A (0.44) PDE2AALDH1A1TSHR
SCHEMBL6680120 0.78 MAPK1 (0.33) PDE2AALDH1A1MAPK1
SCHEMBL12419959 0.78 OPRD1 (0.39) PDE2ATSHRGRIN2B
SCHEMBL8955219 0.78 CA12 (0.35) ALDH1A1TSHRMAPK1TDP1L3MBTL1
SCHEMBL1706121 0.75 PDE2A (0.62) PDE2AAKT1AKT2ALDH1A1TSHR
SCHEMBL13925378 0.75 HIF1A (0.47) PDE2AAKT1AKT2ALDH1A1
SCHEMBL14291912 0.73 PDE2A (0.61) PDE2AAKT1AKT2TSHRGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2940017-B1 Process for making compounds useful as inhibitors of ATR kinase VERTEX PHARMA (US) 2019-08-28 EP disclosed