SCHEMBL21301591

SCHEMBL21301591

CCOC(=O)C(c1ccccc1)N(Cc1cccc(N)c1)C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
HSD17B10 Q99714 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TRPM8 Q7Z2W7 2/20 0.39
OPRK1 P41145 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
BACE1 P56817 5/20 0.38
F10 P00742 1/20 0.37
AKT1 P31749 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
AOC3 Q16853 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16690711 0.92 TRPM8 (0.41) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL8256880 0.90 MEN1 (0.46) TRPM8OPRK1MEN1KMT2ABACE1
SCHEMBL27691292 0.89 TRPM8 (0.41) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL27691293 0.89 TRPM8 (0.41) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL1491418 0.86 ALDH1A1 (0.43) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL1491415 0.86 ALDH1A1 (0.43) ALDH1A1LMNAPOLBHSD17B10L3MBTL1
SCHEMBL14878978 0.84 MEN1 (0.40) TRPM8OPRK1MEN1KMT2ABACE1
SCHEMBL1491639 0.84 CACNA1B (0.39) TRPM8OPRK1BACE1
SCHEMBL1491637 0.84 CACNA1B (0.39) TRPM8OPRK1BACE1
SCHEMBL21301649 0.84 CYP2D6 (0.47) ALDH1A1LMNAPOLBHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3530290-A1 ALPHA AMINOACID ESTER-DRUG CONJUGATES HYDROLYSABLE BY CARBOXYLESTERASE GlaxoSmithKline Intellectual Property Development Limited (GB) 2019-08-28 EP disclosed