SCHEMBL21301649

SCHEMBL21301649

CCOC(=O)C(c1ccccc1)N(Cc1cccc([N+](=O)[O-])c1)C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.47
CYP2C9 P11712 3/20 0.47
CYP2C19 P33261 3/20 0.47
CYP1A2 P05177 1/20 0.47
LMNA P02545 5/20 0.45
ALDH1A1 P00352 4/20 0.45
MAPT P10636 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
MAPK1 P28482 2/20 0.44
ITGA4 P13612 1/20 0.43
ITGB7 P26010 1/20 0.43
OPRK1 P41145 2/20 0.42
RECQL P46063 1/20 0.41
FFAR1 O14842 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.41
HSD17B10 Q99714 1/20 0.41
OPRM1 P35372 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16690714 0.93 CYP2D6 (0.47) CYP2D6CYP2C9CYP2C19CYP1A2LMNA
SCHEMBL14066212 0.92 ITGA4 (0.48) CYP2D6CYP2C9CYP2C19CYP1A2LMNA
SCHEMBL27703141 0.91 CYP2D6 (0.49) CYP2D6CYP2C9CYP2C19CYP1A2LMNA
SCHEMBL27703142 0.91 CYP2D6 (0.49) CYP2D6CYP2C9CYP2C19CYP1A2LMNA
SCHEMBL1491432 0.87 CYP2D6 (0.47) CYP2D6CYP2C9CYP2C19CYP1A2LMNA
SCHEMBL1491427 0.87 CYP2D6 (0.47) CYP2D6CYP2C9CYP2C19CYP1A2LMNA
SCHEMBL1491732 0.85 ALDH1A1 (0.44) CYP2D6CYP2C9CYP2C19CYP1A2LMNA
SCHEMBL1491730 0.85 ALDH1A1 (0.44) CYP2D6CYP2C9CYP2C19CYP1A2LMNA
SCHEMBL21301591 0.84 ALDH1A1 (0.44) LMNAALDH1A1OPRK1L3MBTL1POLB
SCHEMBL6352623 0.82 CYP2D6 (0.45) CYP2D6CYP2C9CYP2C19CYP1A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3530290-A1 ALPHA AMINOACID ESTER-DRUG CONJUGATES HYDROLYSABLE BY CARBOXYLESTERASE GlaxoSmithKline Intellectual Property Development Limited (GB) 2019-08-28 EP disclosed