SCHEMBL21330612

SCHEMBL21330612

Fc1cccc(Oc2ccc(Cl)cc2)n1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
P2RX3 P56373 16/20 0.51
HTT P42858 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8941507 0.85 MEN1 (0.50) MEN1KMT2AP2RX3HTTL3MBTL1
SCHEMBL8941674 0.82 F2 (0.46) HTT
SCHEMBL21330640 0.81 MEN1 (0.48) MEN1KMT2AP2RX3HTTL3MBTL1
SCHEMBL21330627 0.81 MEN1 (0.52) MEN1KMT2AP2RX3HTT
SCHEMBL11684536 0.81 MEN1 (0.47) MEN1KMT2A
SCHEMBL10980485 0.81 HTT (0.47) MEN1KMT2AP2RX3HTTL3MBTL1
SCHEMBL958339 0.81 MEN1 (0.51) MEN1KMT2AP2RX3HTTL3MBTL1
SCHEMBL22061575 0.80 F2 (0.41)
SCHEMBL7228289 0.79 KDM4E (0.47)
SCHEMBL9771157 0.78 HTT (0.47) MEN1KMT2AP2RX3HTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10711006-B2 Selective Bruton's tyrosine kinase inhibitor and use thereof HANGZHOU HERTZ PHARMACEUTICAL CO., LTD. (CN) 2020-07-14 US disclosed
CN-108069974-B Selective Bruton tyrosine kinase inhibitor and application thereof HANGZHOU HERTZ PHARMACEUTICAL CO., LTD. (CN) 2019-12-10 CN disclosed
EP-3543239-A1 SELECTIVE BRUTON'S TYROSINE KINASE INHIBITOR AND USE THEREOF Hangzhou Hertz Pharmaceutical Co., Ltd. (CN) 2019-09-25 EP disclosed
US-20190276461-A1 SELECTIVE BRUTON'S TYROSINE KINASE INHIBITOR AND USE THEREOF Hangzhou Healzen Therapeutics Co., Ltd. (CN) 2019-09-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190276461-A1 SELECTIVE BRUTON'S TYROSINE KINASE INHIBITOR AND USE THEREOF BTK, BMX, KCNK10 MEN1 2111/4885KMT2A 2028/4885P2RX3 947/4885
US-10711006-B2 Selective Bruton's tyrosine kinase inhibitor and use thereof BTK, SYK, LYN MEN1 2441/4885KMT2A 1652/4885P2RX3 1143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.