SCHEMBL21331968

SCHEMBL21331968

COc1ccc(C2CNC(=O)CC2=NO)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.47
CRBN Q96SW2 1/20 0.47
MMP1 P03956 1/20 0.41
MMP13 P45452 1/20 0.41
MAP2K1 Q02750 1/20 0.41
ALDH1A1 P00352 3/20 0.40
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
FPR1 P21462 3/20 0.38
FPR2 P25090 1/20 0.38
TSHR P16473 1/20 0.38
CYP19A1 P11511 1/20 0.37
KDM4E B2RXH2 1/20 0.37
TP53 P04637 1/20 0.37
RAB9A P51151 1/20 0.37
MAP2K3 P46734 1/20 0.37
POLB P06746 1/20 0.37
RECQL P46063 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21331966 1.00 DDB1 (0.47) DDB1CRBNMMP1MMP13MAP2K1
SCHEMBL21332020 0.82 DDB1 (0.51) DDB1CRBNMMP1MMP13MAP2K1
SCHEMBL21331977 0.79 FPR1 (0.46) ALDH1A1FPR1FPR2KMT2A
SCHEMBL21331979 0.79 FPR1 (0.46) ALDH1A1FPR1FPR2KMT2A
SCHEMBL21332358 0.77 FPR1 (0.41) FPR1FPR2
SCHEMBL21332359 0.77 FPR1 (0.41) FPR1FPR2
SCHEMBL8530171 0.72 DDB1 (0.44) DDB1CRBNMMP1MMP13MAP2K1
SCHEMBL8530170 0.72 DDB1 (0.44) DDB1CRBNMMP1MMP13MAP2K1
SCHEMBL1268717 0.69 TSHR (0.69) MAP2K1ALDH1A1ALOX15TSHRKDM4E
SCHEMBL18117753 0.69 TSHR (0.69) MAP2K1ALDH1A1ALOX15TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170904-A1 PIPERIDINES OR PIPERIDONES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-09-12 WO disclosed