SCHEMBL21332020

SCHEMBL21332020

COc1ccc(C2CNC(=O)CC2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.51
CRBN Q96SW2 1/20 0.51
MAP2K1 Q02750 1/20 0.44
MMP1 P03956 1/20 0.42
MMP13 P45452 1/20 0.42
TSHR P16473 2/20 0.41
ALDH1A1 P00352 2/20 0.40
CYP19A1 P11511 1/20 0.40
MAP2K3 P46734 1/20 0.40
PDE4A P27815 3/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
MAOA P21397 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21331966 0.82 DDB1 (0.47) DDB1CRBNMAP2K1MMP1MMP13
SCHEMBL21331968 0.82 DDB1 (0.47) DDB1CRBNMAP2K1MMP1MMP13
SCHEMBL4768818 0.78 DDB1 (0.44) DDB1CRBNTSHRCYP19A1GAA
SCHEMBL21332230 0.74 FPR1 (0.44)
SCHEMBL18117753 0.73 TSHR (0.69) MAP2K1TSHRALDH1A1PDE4APDE4B
SCHEMBL1268717 0.73 TSHR (0.69) MAP2K1TSHRALDH1A1PDE4APDE4B
SCHEMBL9537344 0.72 DDB1 (0.56) DDB1CRBNMMP1MMP13ALDH1A1
SCHEMBL27965543 0.70 CRBN (0.71) DDB1CRBNMMP1MMP13TSHR
SCHEMBL19972309 0.69 KDM1A (0.56) DDB1CRBNMAP2K1TSHRPDE4A
SCHEMBL19985875 0.69 KDM1A (0.56) DDB1CRBNMAP2K1TSHRPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170904-A1 PIPERIDINES OR PIPERIDONES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-09-12 WO disclosed
WO-2019170904-A1 PIPERIDINES OR PIPERIDONES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-09-12 WO disclosed