SCHEMBL21332885

SCHEMBL21332885

Cc1c(C(=O)Cn2cc(Br)ccc2=O)cnn1Cc1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 7/20 0.41
S1PR2 O95136 1/20 0.39
POLB P06746 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
MITF O75030 2/20 0.39
HTT P42858 2/20 0.39
RAB9A P51151 2/20 0.39
PKM P14618 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TP53 P04637 1/20 0.37
SLC2A1 P11166 1/20 0.37
SLC2A3 P11169 1/20 0.37
TRPV4 Q9HBA0 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CREBBP Q92793 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21332946 0.89 S1PR2 (0.47) PTGDR2S1PR2POLBRAB9ATP53
SCHEMBL21332838 0.85 PTGDR2 (0.41) PTGDR2S1PR2POLBMITFHTT
SCHEMBL21333280 0.84 KDM4E (0.39) PTGDR2S1PR2RAB9APKMKDM4E
SCHEMBL21333089 0.82 PTGDR2 (0.39) PTGDR2S1PR2POLBMITFHTT
SCHEMBL21333289 0.82 S1PR2 (0.43) PTGDR2S1PR2RAB9ATP53KDM4E
SCHEMBL30866465 0.81 KMT2A (0.42) PTGDR2S1PR2POLBTDP1HTT
SCHEMBL21333435 0.81 KMT2A (0.42) PTGDR2S1PR2POLBTDP1HTT
SCHEMBL21333112 0.80 S1PR2 (0.61) PTGDR2S1PR2MITFHTTRAB9A
SCHEMBL30866453 0.80 CREBBP (0.43) PTGDR2S1PR2SLC2A1SLC2A3SMN1; SMN2
SCHEMBL21333412 0.79 PTGER1 (0.48) PTGDR2POLBTDP1TP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3762377-B1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND MEDICAL USES THEREOF UNIV CORNELL (US) 2025-08-20 EP disclosed
US-11964960-B2 Pyridinone- and pyridazinone-based compounds and uses thereof CORNELL UNIVERSITY (US) 2024-04-23 US disclosed
EP-3762377-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND MEDICAL USES THEREOF Cook, Timothy, H. (US) 2021-01-13 EP disclosed
US-20200407339-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND USES THEREOF TRI-INSTITUTIONAL THERAPEUTICS DISCOVERY INSTITUTE 2020-12-31 US disclosed
US-20200407339-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND USES THEREOF TRI-INSTITUTIONAL THERAPEUTICS DISCOVERY INSTITUTE 2020-12-31 US disclosed
WO-2019173790-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND MEDICAL USES THEREOF HLA TIMOTHY (US) 2019-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200407339-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND USES THEREOF PTGER1, LOXL1, COL1A1 PTGDR2 103/4885S1PR2 601/4885POLB 3175/4885
US-11964960-B2 Pyridinone- and pyridazinone-based compounds and uses thereof PTGER1, LOXL1, COL1A1 PTGDR2 103/4885S1PR2 601/4885POLB 3175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.