SCHEMBL21336611

SCHEMBL21336611

CCCC(C)c1ccc(C#N)cc1C

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.36
CRHR1 P34998 2/20 0.35
ALDH1A1 P00352 1/20 0.35
SLC6A3 Q01959 1/20 0.35
TRPV4 Q9HBA0 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
S1PR1 P21453 2/20 0.33
FFAR1 O14842 1/20 0.33
GLA P06280 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32
DRD2 P14416 2/20 0.32
DRD3 P35462 2/20 0.32
HCAR2 Q8TDS4 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19464642 0.86 CYP2A6 (0.38) CYP2A6CRHR1ALDH1A1TRPV4S1PR1
SCHEMBL20963140 0.82 AR (0.37) CYP2A6CRHR1SLC6A3TRPV4MEN1
SCHEMBL18552786 0.82 CYP2A6 (0.35) CYP2A6SLC6A3TRPV4MEN1KMT2A
SCHEMBL24767625 0.82 MEN1 (0.35) CYP2A6ALDH1A1SLC6A3TRPV4MEN1
SCHEMBL28248925 0.80 CYP2A6 (0.44) CYP2A6ALDH1A1GLAESR1ESR2
SCHEMBL22796684 0.80 AR (0.42) TRPV4AR
SCHEMBL19068977 0.79 SCN1A (0.40) CYP2A6SLC6A3TRPV4MEN1KMT2A
SCHEMBL21725516 0.78 TRPV4 (0.42) ALDH1A1TRPV4GLAAR
SCHEMBL105403 0.78 ALDH1A1 (0.43) CYP2A6ALDH1A1GLAAR
SCHEMBL19987487 0.77 CRHR1 (0.42) CYP2A6CRHR1ALDH1A1TRPV4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed