SCHEMBL21336724

SCHEMBL21336724

CC1CN(c2ccc(C(=O)OCc3ccccc3)cn2)CC(C)N1C(=O)CN

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 10/20 0.51
HDAC2 Q92769 2/20 0.51
HDAC3 O15379 1/20 0.51
CYP2C9 P11712 1/20 0.51
SLC6A4 P31645 1/20 0.51
SLC6A3 Q01959 1/20 0.51
MAPKAPK3 Q16644 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
SGPL1 O95470 1/20 0.47
KMT2A Q03164 3/20 0.43
MEN1 O00255 1/20 0.43
RAB9A P51151 4/20 0.43
NPC1 O15118 3/20 0.43
P2RY12 Q9H244 1/20 0.43
LMNA P02545 3/20 0.42
TDP1 Q9NUW8 1/20 0.42
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21336665 0.82 KMT2A (0.48) HDAC1HDAC2HDAC3CYP2C9SLC6A4
SCHEMBL12542345 0.78 SGPL1 (0.54) HDAC1HDAC2HDAC3CYP2C9SLC6A4
SCHEMBL23183064 0.76 KMT2A (0.57) HDAC1SLC6A3KMT2AMEN1RAB9A
SCHEMBL18436101 0.76 HSD11B1 (0.43)
SCHEMBL18436778 0.76 HSD11B1 (0.43)
SCHEMBL18436960 0.75 HSD11B1 (0.42) HDAC1
SCHEMBL8241566 0.74 HDAC1 (0.72) HDAC1HDAC2HDAC3CYP2C9SLC6A4
SCHEMBL19581104 0.74 KMT2A (0.55) HDAC1HDAC2HDAC3CYP2C9SLC6A4
SCHEMBL17128146 0.74 RAB9A (0.52) HDAC1SGPL1KMT2ARAB9ANPC1
SCHEMBL19580906 0.74 KMT2A (0.52) HDAC1HDAC2HDAC3CYP2C9SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed