SCHEMBL21336795

SCHEMBL21336795

COc1c(NCCNc2ccc(C(C)(C)O)cn2)cnc2c(-c3ccc(C#N)cc3)cccc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.33
NTRK3 Q16288 1/20 0.33
NTRK2 Q16620 1/20 0.33
TTK P33981 1/20 0.32
DPP4 P27487 3/20 0.32
SLC22A12 Q96S37 1/20 0.32
TYK2 P29597 4/20 0.31
JAK1 P23458 1/20 0.31
STAT3 P40763 1/20 0.31
KCNH2 Q12809 1/20 0.31
CNR2 P34972 1/20 0.31
KDM4A O75164 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
GSK3B P49841 1/20 0.31
SGK1 O00141 1/20 0.31
MAPK1 P28482 1/20 0.31
HTR1A P08908 1/20 0.30
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21336578 0.88 TTK (0.32) NTRK1NTRK3NTRK2TTKSLC22A12
SCHEMBL18436403 0.87 EGLN1 (0.34) SLC22A12MAPK14EGLN1
SCHEMBL18436267 0.86 DPP4 (0.34) DPP4SLC22A12CNR2KDM4AKDM5B
SCHEMBL18436867 0.86 ENPP1 (0.34) NTRK1NTRK3NTRK2TTKTYK2
SCHEMBL18436916 0.85 DPP4 (0.34) DPP4KDM1A
SCHEMBL18436758 0.84 KDM1A (0.34) NTRK1NTRK3NTRK2TYK2MAPK1
SCHEMBL21336708 0.83 HTR1A (0.36) SLC22A12STAT3KDM4AKDM5BHTR1A
SCHEMBL18436682 0.81 RAD52 (0.38) SLC22A12STAT3KDM4AKDM5BHTR1A
SCHEMBL18436729 0.81 CD274 (0.43) KDM4AKDM5BMAPK1EGLN1
SCHEMBL18436930 0.79 POLB (0.39) CNR2KDM4AKDM5BHTR1AEGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed