SCHEMBL21337488

SCHEMBL21337488

CCC(C)N(CC1(N2CCN(Cc3ccccc3)CC2)CC1)c1ccccn1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 18/20 0.64
OPRM1 P35372 17/20 0.64
KCNH2 Q12809 8/20 0.47
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21337250 0.85 SIGMAR1 (0.48) SIGMAR1OPRM1
SCHEMBL21337586 0.78 SIGMAR1 (0.62) SIGMAR1OPRM1KCNH2
SCHEMBL18458660 0.78 OPRM1 (1.00) SIGMAR1OPRM1KCNH2
SCHEMBL21337397 0.73 SIGMAR1 (0.50) SIGMAR1OPRM1KCNH2
SCHEMBL18426780 0.73 SIGMAR1 (0.87) SIGMAR1OPRM1KCNH2
SCHEMBL22445667 0.72 SIGMAR1 (0.62) SIGMAR1OPRM1KCNH2ACHE
SCHEMBL18458977 0.71 SIGMAR1 (0.54) SIGMAR1OPRM1KCNH2
SCHEMBL21337445 0.71 SIGMAR1 (0.52) SIGMAR1OPRM1KCNH2
SCHEMBL18425865 0.71 SIGMAR1 (0.68) SIGMAR1OPRM1KCNH2
SCHEMBL20599284 0.71 OPRM1 (0.69) SIGMAR1OPRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3328853-B1 SUBSTITUTED AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS SA (ES) 2019-09-11 EP disclosed