SCHEMBL21337397

SCHEMBL21337397

CCC(O)N(CC1(N2CCN(Cc3ccccc3)CC2)CC1)c1ccc(C(F)(F)F)cn1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 17/20 0.50
OPRM1 P35372 16/20 0.50
KCNH2 Q12809 7/20 0.50
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
CHRM4 P08173 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18426014 0.82 SIGMAR1 (0.72) SIGMAR1OPRM1KCNH2
SCHEMBL21337398 0.82 SIGMAR1 (0.54) SIGMAR1OPRM1KCNH2CHRM4
SCHEMBL18458556 0.78 SIGMAR1 (0.71) SIGMAR1OPRM1KCNH2
SCHEMBL18426659 0.77 SIGMAR1 (0.73) SIGMAR1OPRM1KCNH2
SCHEMBL18458019 0.75 SIGMAR1 (0.62) SIGMAR1OPRM1KCNH2
SCHEMBL21337488 0.73 SIGMAR1 (0.64) SIGMAR1OPRM1KCNH2
SCHEMBL18458499 0.73 ACHE (0.47) SIGMAR1OPRM1KCNH2POLBGAA
SCHEMBL20621716 0.72 SIGMAR1 (0.48) SIGMAR1OPRM1KCNH2
SCHEMBL21337445 0.72 SIGMAR1 (0.52) SIGMAR1OPRM1KCNH2POLB
SCHEMBL18426860 0.70 SIGMAR1 (0.76) SIGMAR1OPRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3328853-B1 SUBSTITUTED AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS SA (ES) 2019-09-11 EP disclosed