SCHEMBL21340862

SCHEMBL21340862

CC1CC(NC(=O)OC(C)(C)C)C(=O)N1c1ccc(-c2ccccc2P(C)C)c(F)c1F

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FPR1 P21462 19/20 0.49
FPR2 P25090 19/20 0.49
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24337033 0.87 FPR2 (0.65) FPR1FPR2
SCHEMBL21319266 0.87 FPR2 (0.65) FPR1FPR2
SCHEMBL30832912 0.87 FPR2 (0.65) FPR1FPR2
SCHEMBL24093591 0.84 FPR2 (0.48) FPR1FPR2
SCHEMBL25712974 0.81 FPR2 (0.49) FPR1FPR2
SCHEMBL24093677 0.80 FPR2 (0.46) FPR1FPR2
SCHEMBL21341184 0.80 FPR1 (0.41) FPR1FPR2HDAC1HDAC8HDAC6
SCHEMBL30832910 0.80 FPR1 (0.41) FPR1FPR2HDAC1HDAC8HDAC6
SCHEMBL24093594 0.79 FPR1 (0.79) FPR1FPR2
SCHEMBL24093581 0.77 FPR1 (0.52) FPR1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3981767-A1 PHENYLPYRROLIDINONE FORMYL PEPTIDE 2 RECEPTOR AGONISTS Bristol-Myers Squibb Company (US) 2022-04-13 EP disclosed
EP-3762380-B1 PHENYLPYRROLIDINONE FORMYL PEPTIDE 2 RECEPTOR AGONISTS BRISTOL MYERS SQUIBB CO (US) 2021-12-15 EP disclosed
WO-2019173182-A1 PHENYLPYRROLIDINONE FORMYL PEPTIDE 2 RECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2019-09-12 WO disclosed