SCHEMBL21345488

SCHEMBL21345488

Oc1cc2c(cc1O)C1(c3ccccc3N2c2ccccc2)c2ccccc2N(c2ccccc2)c2cc(O)c(O)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 1/20 0.38
ALDH1A1 P00352 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
THPO P40225 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
MAPK1 P28482 1/20 0.34
IDH1 O75874 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ESR1 P03372 1/20 0.33
SRC P12931 2/20 0.32
FGFR1 P11362 1/20 0.32
NPSR1 Q6W5P4 2/20 0.32
CES2 O00748 1/20 0.32
BCHE P06276 1/20 0.32
GAA P10253 1/20 0.32
CES1 P23141 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21345468 0.90 ESR1 (0.35) ADAMTS5ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL20202064 0.84 ALDH1A1 (0.44) ADAMTS5ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL21345469 0.80 PGR (0.37) ALDH1A1ESR1PGR
SCHEMBL12723310 0.79 ALDH1A1 (0.37) ADAMTS5ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL2754774 0.77 GAA (0.44) ADAMTS5ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL29776217 0.77 GAA (0.44) ADAMTS5ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL21350687 0.76 PSMB1 (0.36) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL18387369 0.76 CNR1 (0.40) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL17657227 0.76 CNR1 (0.40) ADAMTS5ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL3199631 0.76 EGLN1 (0.36) ADAMTS5ALDH1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10953369-B2 Spirocentric compounds and polymers thereof GEORGIA TECH RESEARCH CORPORATION (US) 2021-03-23 US disclosed
US-20190276454-A1 Spirocentric Compounds and Polymers Thereof GEORGIA TECH RESEARCH CORPORATION 2019-09-12 US disclosed
WO-2019173646-A1 SPIROCENTRIC COMPOUNDS AND POLYMERS THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190276454-A1 Spirocentric Compounds and Polymers Thereof PKD1, PKD2, VIM ADAMTS5 2049/4885ALDH1A1 2886/4885CYP1A2 4805/4885
US-10953369-B2 Spirocentric compounds and polymers thereof PKD1, PKD2, VIM ADAMTS5 2049/4885ALDH1A1 2886/4885CYP1A2 4805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.