SCHEMBL2134679

SCHEMBL2134679

O=C(Cc1ccccn1)Nc1cccc(Cl)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.67
MAPT P10636 2/20 0.67
NPC1 O15118 1/20 0.67
GRM4 Q14833 1/20 0.63
HDAC6 Q9UBN7 1/20 0.63
ALDH1A1 P00352 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2C19 P33261 1/20 0.61
KCNJ5 P48544 1/20 0.60
KCNJ3 P48549 1/20 0.60
LMNA P02545 1/20 0.58
KDR P35968 1/20 0.58
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA5A P35218 1/20 0.55
CA7 P43166 1/20 0.55
CA5B Q9Y2D0 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3453018 0.84 CA1 (0.67) RAB9ANPC1ALDH1A1LMNAMEN1
SCHEMBL2028409 0.84 CA1 (0.69) RAB9ANPC1HDAC6LMNAMEN1
SCHEMBL259393 0.83 NPC1 (0.67) RAB9ANPC1ALDH1A1CYP1A2CYP3A4
SCHEMBL31240480 0.81 GSK3A (0.63) RAB9AMAPTNPC1MEN1KMT2A
SCHEMBL6436243 0.81 CA1 (0.59) RAB9AMAPTNPC1ALDH1A1MEN1
SCHEMBL6931979 0.79 F2 (0.58) RAB9AMAPTNPC1GRM4HDAC6
SCHEMBL10576461 0.78 CA1 (0.67) RAB9AMAPTNPC1HDAC6ALDH1A1
SCHEMBL11617075 0.78 SMN1; SMN2 (0.62) RAB9AMAPTNPC1GRM4HDAC6
SCHEMBL2530324 0.78 GRM4 (1.00) RAB9ANPC1GRM4HDAC6KDR
SCHEMBL11531211 0.78 KMT2A (0.76) RAB9AMAPTNPC1ALDH1A1KCNJ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9463187-B2 Methylphenidate derivatives and uses of them AMPIO PHARMACEUTICALS, INC. (US) 2016-10-11 US disclosed
US-20120101129-A1 Methylphenidate Derivatives and Uses of Them AMPIO PHARMACEUTICALS, INC. 2012-04-26 US disclosed
US-8076485-B2 Methylphenidate derivatives and uses of them INSTITUTE FOR MOLECULAR MEDICINE, INC. (US) 2011-12-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120101129-A1 Methylphenidate Derivatives and Uses of Them SLC6A3, COMT, UGT1A1 RAB9A 1329/4885MAPT 1011/4885NPC1 390/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.