SCHEMBL21362446

SCHEMBL21362446

CC[S+]([O-])Cc1ccc(C(=O)c2ccc(OC)c(F)c2)c(-c2cn(C)c(=O)cc2[C@H](C)NS)c1

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.36
ACHE P22303 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158057 1.00 BRD4 (0.36) BRD4ACHETAS1R3TAS1R1
SCHEMBL20157434 0.79 BRD4 (0.33) BRD4
SCHEMBL21362138 0.79 BRD4 (0.38) BRD4ACHETAS1R3TAS1R1
SCHEMBL21362238 0.78 BRD4 (0.37) BRD4ACHETAS1R3TAS1R1
SCHEMBL21362057 0.78 MAPK14 (0.32) BRD4
SCHEMBL21362147 0.76 BRD4 (0.31) BRD4
SCHEMBL21352136 0.76 BRD4 (0.38) BRD4ACHETAS1R3TAS1R1
SCHEMBL21564841 0.75 DRD4 (0.32) BRD4
SCHEMBL20157926 0.73 BRD4 (0.37) BRD4
SCHEMBL20157431 0.73 THRB (0.34) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed