SCHEMBL21362535

SCHEMBL21362535

C=C(c1ccc(F)cc1)c1cc(Cl)c(NC(=O)OC(C)(C)C)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 2/20 0.43
KCNQ4 P56696 3/20 0.38
KCNQ5 Q9NR82 3/20 0.38
CYP17A1 P05093 1/20 0.37
KDM4E B2RXH2 2/20 0.37
RAB9A P51151 3/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
NPY1R P25929 1/20 0.36
NPY2R P49146 1/20 0.36
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
NPC1 O15118 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
RXRA P19793 1/20 0.34
ATR Q13535 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157868 0.89 SMN1; SMN2 (0.45) SMN1; SMN2ALDH1A1HPGDKCNQ4KCNQ5
SCHEMBL21564978 0.89 ALDH1A1 (0.39) SMN1; SMN2ALDH1A1HPGDKCNQ4KCNQ5
SCHEMBL21564976 0.81 KCNQ4 (0.39) SMN1; SMN2ALDH1A1HPGDKCNQ4KCNQ5
SCHEMBL20158012 0.80 PPARG (0.40) SMN1; SMN2ALDH1A1HPGDKDM4ERAB9A
SCHEMBL20157982 0.79 LCK (0.39) SMN1; SMN2ALDH1A1HPGDKDM4ERAB9A
SCHEMBL21362424 0.76 SMN1; SMN2 (0.40) SMN1; SMN2ALDH1A1HPGDCYP17A1KDM4E
SCHEMBL29840249 0.75 AAK1 (0.46) KCNQ4KCNQ5CYP17A1RAB9ALMNA
SCHEMBL28190043 0.74 CA12 (0.40) RAB9ACA12CA1CA2CA9
SCHEMBL30947444 0.72 CYP17A1 (0.42) KCNQ4KCNQ5CYP17A1RAB9ACA12
SCHEMBL29236468 0.72 CYP17A1 (0.42) KCNQ4KCNQ5CYP17A1RAB9ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed