SCHEMBL21362424

SCHEMBL21362424

CCc1ccc(C(=O)c2cc(Cl)c(NC(=O)OC(C)(C)C)cc2Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.40
RAB9A P51151 3/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 3/20 0.39
MAPT P10636 5/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
NPY1R P25929 1/20 0.38
NPY2R P49146 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
HTT P42858 1/20 0.38
MKNK2 Q9HBH9 1/20 0.36
EGFR P00533 1/20 0.36
AGTR1 P30556 1/20 0.36
CYP17A1 P05093 1/20 0.36
ATR Q13535 1/20 0.36
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158012 0.89 PPARG (0.40) SMN1; SMN2RAB9ANPC1MAPTALDH1A1
SCHEMBL20157982 0.88 LCK (0.39) SMN1; SMN2RAB9ANPC1MAPTALDH1A1
SCHEMBL20157868 0.87 SMN1; SMN2 (0.45) SMN1; SMN2RAB9ANPC1MAPTALDH1A1
SCHEMBL21564976 0.77 KCNQ4 (0.39) SMN1; SMN2NPC1GAAALDH1A1LMNA
SCHEMBL21362535 0.76 SMN1; SMN2 (0.43) SMN1; SMN2RAB9ANPC1MAPTALDH1A1
SCHEMBL3682780 0.74 MAPT (0.44) SMN1; SMN2RAB9ANPC1GAAMAPT
SCHEMBL21362622 0.74 MAPT (0.46) SMN1; SMN2RAB9ANPC1GAAMAPT
SCHEMBL28190043 0.74 CA12 (0.40) RAB9ANPC1HTTATRCA12
SCHEMBL21564978 0.72 ALDH1A1 (0.39) SMN1; SMN2RAB9AMAPTALDH1A1KDM4E
SCHEMBL8258036 0.71 SLC10A6 (0.50) SMN1; SMN2GAAMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed