SCHEMBL21362561

SCHEMBL21362561

CNc1c[nH]c(C(N)=O)c1C

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCNC P24863 6/20 0.46
CDK8 P49336 6/20 0.46
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
GDA Q9Y2T3 1/20 0.33
NNMT P40261 2/20 0.32
MAP2K3 P46734 1/20 0.31
MAPK14 Q16539 1/20 0.31
IKBKB O14920 1/20 0.30
ACHE P22303 1/20 0.30
PRKCI P41743 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157257 0.75 CCNC (0.51) CCNCCDK8ALDH1A1KDM4EGDA
SCHEMBL7560908 0.74 CCNC (0.50) CCNCCDK8ALDH1A1KDM4EGDA
SCHEMBL7116182 0.71 CCNC (0.47) CCNCCDK8ALDH1A1KDM4E
SCHEMBL30317801 0.68 CCNC (0.45) CCNCCDK8GDA
SCHEMBL19332726 0.67 CCNC (0.44) CCNCCDK8ALDH1A1KDM4E
SCHEMBL7475587 0.65 CCNC (0.42) CCNCCDK8ALDH1A1KDM4EGDA
SCHEMBL23863591 0.65 PDPK1 (0.55) ALDH1A1KDM4EGLAGAANNMT
SCHEMBL3138229 0.65 GRM1 (0.49) CCNCCDK8ALDH1A1
SCHEMBL8537859 0.64 KDM4E (0.39) ALDH1A1KDM4EGLAGAANNMT
SCHEMBL16116379 0.63 CCNC (1.00) CCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed