SCHEMBL21362629

SCHEMBL21362629

CCc1cc(CO)c(Br)cc1C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 1/20 0.36
PGK2 P07205 1/20 0.36
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
SHBG P04278 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
ALDH1A1 P00352 1/20 0.30
THRB P10828 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3958466 0.82 SHBG (0.39) SHBGLMNATSHRNPSR1ALOX15
SCHEMBL6828121 0.80 SHBG (0.38) SHBGTSHRHPGDALOX15ALOX12
SCHEMBL1318936 0.80 SHBG (0.42) PGK1PGK2SHBGNPSR1ALOX15
SCHEMBL17244913 0.78 ALDH1A1 (0.39) PGK1PGK2NOS3NOS1NOS2
SCHEMBL29613199 0.76 SHBG (0.42) PGK1PGK2SHBGHPGDNPSR1
SCHEMBL17244912 0.76 SHBG (0.42) PGK1PGK2SHBGHPGDNPSR1
SCHEMBL6745128 0.75 KDM1A (0.38) SHBGNPSR1ALOX15ALOX12ALDH1A1
SCHEMBL20157706 0.75 CD44 (0.37) SHBGLMNAALOX15ALOX12
SCHEMBL15788771 0.75 TSHR (0.44) NOS3NOS1NOS2LMNATSHR
SCHEMBL26036108 0.74 PDGFRB (0.40) HPGDALDH1A1THRBIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed