SCHEMBL21362785

SCHEMBL21362785

CCNSc1ccc(C(O)c2ccc(F)cc2)c(Br)c1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
F2RL1 P55085 3/20 0.30
AOC3 Q16853 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11867787 0.75 HDAC3 (0.36) KMT2ATHRATHRBBRD4AOC3
SCHEMBL21362648 0.73 ACHE (0.39) KMT2ATHRATHRBBRD4CREBBP
SCHEMBL20157454 0.72 ALDH1A1 (0.46) KMT2AMEN1
SCHEMBL20157912 0.72 BRD4 (0.32) KMT2AMEN1THRATHRBBRD4
SCHEMBL20157878 0.72 CHRNA7 (0.38) KMT2A
SCHEMBL11857823 0.71 APLNR (0.44) KMT2AMEN1THRATHRB
SCHEMBL20154947 0.68 EPAS1 (0.45) BRD4
SCHEMBL21564724 0.67 HPGD (0.40) KMT2A
SCHEMBL11853713 0.67 IDO1 (0.41) KMT2AMEN1
SCHEMBL21352143 0.66 BRD4 (0.34) ALOX5KMT2ATHRATHRBBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed