SCHEMBL21384575

SCHEMBL21384575

O=S(=O)(Nc1ccc(Cl)cc1Nc1ccc(C(F)(F)F)cc1Cl)C1CC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.46
MRGPRX1 Q96LB2 2/20 0.43
KIF11 P52732 1/20 0.41
CNR2 P34972 7/20 0.41
CNR1 P21554 3/20 0.41
DDR1 Q08345 1/20 0.41
IDH1 O75874 1/20 0.40
CHRNA7 P36544 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CCR2 P41597 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384560 0.95 MCL1 (0.46) MCL1MRGPRX1KIF11CNR2CNR1
SCHEMBL21384550 0.90 MCL1 (0.44) MCL1MRGPRX1KIF11CNR2CNR1
SCHEMBL21384576 0.81 MRGPRX1 (0.63) MRGPRX1IDH1CA12CA1CA2
SCHEMBL21394361 0.76 MRGPRX1 (0.58) MRGPRX1IDH1CA12CA1CA2
SCHEMBL393515 0.74 BRAF (0.40) MRGPRX1CNR2CNR1CCR2
SCHEMBL21394560 0.74 MRGPRX1 (0.51) MRGPRX1CA12CA1CA2CA9
SCHEMBL21394420 0.74 MRGPRX1 (0.56) MRGPRX1CA12CA1CA2CA9
SCHEMBL21394417 0.74 MRGPRX1 (0.53) MRGPRX1CA12CA1CA2CA9
SCHEMBL21381357 0.73 MAPT (0.48) MCL1KIF11CHRNA7CA12CA1
SCHEMBL21381353 0.73 MRGPRX1 (0.62) MRGPRX1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed